Tirzepatide ni munkhwala uphya uwo ukupokelera viŵaro viŵiri, uwo sono ukugwiriskirika nchito chomene pa vinthu ivi:
1. Kututuwa chomene/kulongozga kwakujumphizga
Ivyo vikupangiska:
Iwo ukukhozgera kuchepeska thupi mwa kukanizga chakurya, kuchedweska kufunyapo kanthu kwa m’mimba, kuchepeskako vyakurya vya calorie.
Iwo ukugwira ntchito chomene kuluska munkhwala wa GLP-1 wa chikhalidwe (nga ni semaglutide).
Vinthu vyakukhwaskana na chipatala:
Mndandanda wa SURMOUNT wa mayesero ukalongora kuti pafupifupi kuthukira kwa ŵalwari ŵakunenepa (kwambura shuga) kukaŵa:
15%-20% (5 mg / sabata)
20%-22% (10-15 mg / sabata)
Vimanyikwiro vyakuwoneka makora nga ni chiuno, mafuta gha ndopa, na kuthamanga kwa ndopa.
Viŵelengelo vyakugwiriskira ntchito:
Obese (BMI Great kuluska panji yakuyana waka na 30 kg / m2) panji kulemera chomene (BMI Greater kuluska panji yakuyana waka na 27 kg / m2) na pafupifupi kututuwa kumoza - pakuyaniska matenda (nga ni hypertension, mtundu wachiŵiri wa shuga, dyslipidemia).
2.2 mtundu wa shuga wa shuga wa mtundu wa 1.2 matenda gha shuga 1.2 1, 1.2 matenda gha 1.2 at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at at 1.2 matenda gha shuga pa 1.2 matenda gha shuga 1.2 pa 1.2 matenda gha shuga 1.2 matenda 1.2 matenda gha shuga 1.2 matenda 1.2 matenda gha shuga 1.2 matenda 1..
Ivyo vikupangiska:
Nga ni umo vikuŵira na vyakurya na maseŵero ghakukhozga thupi, vikupangiska kuti shuga wa mu ndopa waŵe na suzgo la shuga mu ndopa.
Iwo ukupangiska GIP na GLP-1 receptors, vikupangiska kuti insulini yiŵe yiwemi, yikukanizga glucagon, na kucedweska kufwatuka kwa m’mimba, mwakuti yichepeskenge kuziŵizga kurya na shuga wa ndopa.
Vinthu vyakukhwaskana na chipatala:
Kuchepeska chomene HbA1c (hemoglobin ya glycosylated) na 1.8%-2.4%.
Ŵalwari ŵanyake ŵangakwaniska kuchepeskeka kwa thupi pa nyengo ya kuchizgika (kusazgirapo kwakusazgikira).
Viŵelengelo vyakugwiriskira ntchito:
Ŵalwari ŵalara awo ŵali na suzgo la shuga la mtundu wa 2, chomenechomene awo ŵali na suzgo la kunenepa chomene panji ŵakunenepa chomene pamoza na suzgo la shuga.
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